Small-molecule modulators of serine protease inhibitor proteins (serpins)
Tahsin F. Kellici, E. Pilka, Michael J. Bodkin
Topics & Concepts
Drug discoverySerpinSerine proteaseIn silicoComputational biologySmall moleculeDrug designProteaseRational designBiologyBioinformaticsBiochemistryEnzymeGeneticsGeneProtease and Inhibitor MechanismsBlood Coagulation and Thrombosis MechanismsProtein Kinase Regulation and GTPase Signaling