Novel potent SOS1 inhibitors containing a tricyclic quinazoline scaffold: A joint view of experiments and simulations
Luolong Qing, Zhengzai Cheng, Juan Xu, Ziwei Wang, Yuanyuan Li, Mario Gauthier, Silong Zhang, Huan He
Topics & Concepts
ChemistryTricyclicQuinazolineScaffoldStereochemistryPharmacologyCombinatorial chemistryBiomedical engineeringMedicineQuinazolinone synthesis and applicationsSynthesis and biological activitySynthesis and Characterization of Heterocyclic Compounds