Discovery of high-affinity ligands for prostatic acid phosphatase via DNA-encoded library screening enables targeted cancer therapy
Tony Georgiev, Francesca Migliorini, Andrea Ciamarone, Marco Müller, Ilaria Biancofiore, Pinuccia Faviana, Francesco Bartoli, Y Kim, Lucrezia Principi, Ettore Gilardoni, Gabriele Bassi, Nicholas Favalli, Emanuele Puca, Dario Neri, Sebastian Oehler, Samuele Cazzamalli
Topics & Concepts
Prostatic acid phosphataseDNACancerCancer researchCancer therapyChemistryProstate cancerPhosphataseBiochemistryComputational biologyMolecular biologyMedicineBiologyEnzymeInternal medicinePeptidase Inhibition and AnalysisBiochemical and Molecular ResearchGlycosylation and Glycoproteins Research