Litcius/Paper detail

Selection of DNA-encoded chemical libraries against endogenous membrane proteins on live cells

Yiran Huang, Ling Meng, Qigui Nie, Yu Zhou, Langdong Chen, Shilian Yang, Yi Man Eva Fung, Xiaomeng Li, Cen Huang, Yan Cao, Yizhou Li, Xiaoyu Li

2020Nature Chemistry142 citationsDOI

Topics & Concepts

Drug discoveryMembrane proteinChemistryDNAChemical biologyHigh-throughput screeningChemical libraryComputational biologyFunction (biology)Ligand (biochemistry)Integral membrane proteinMembraneBiochemistryCell biologyReceptorBiologySmall moleculeAdvanced biosensing and bioanalysis techniquesChemical Synthesis and AnalysisClick Chemistry and Applications