Phenotype Screening of an Azole-bisindole Chemical Library Identifies URB1483 as a New Antileishmanial Agent Devoid of Toxicity on Human Cells
Aurora Diotallevi, Laura Scalvini, Gloria Buffi, Yolanda Pérez‐Pertejo, Mauro De Santi, Michele Verboni, Gianfranco Favi, Mauro Magnani, Alessio Lodola, Simone Lucarini, Luca Galluzzi
Abstract
emerges as a new anti-infective agent with remarkable antileishmanial activity and no cytotoxic effects on human and canine cells.
Topics & Concepts
Leishmania infantumAmastigoteHaCaTCytotoxicityIn vitroIntracellularPharmacologyLeishmaniasisToxicityCell cultureChemistryLeishmaniaBiologyIC50ImmunologyVisceral leishmaniasisBiochemistryParasite hostingGeneticsComputer scienceOrganic chemistryWorld Wide WebResearch on Leishmaniasis StudiesCancer therapeutics and mechanismsTrypanosoma species research and implications