Harnessing systematic protein–ligand interaction fingerprints for drug discovery
Zheng Zhao, Philip E. Bourne
Topics & Concepts
KinomeDrug discoveryComputational biologyAllosteric regulationProteomeDrugProtein–protein interactionLigand (biochemistry)Protein ligandDrug developmentLigand efficiencyDruggabilityChemistryBiologyBioinformaticsKinasePharmacologyBiochemistryReceptorGeneComputational Drug Discovery MethodsMicrobial Natural Products and BiosynthesisPharmacogenetics and Drug Metabolism