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Seeking Nonspecific Binding: Assessing the Reliability of Tissue Dilutions for Calculating Fraction Unbound

William J. Jusko, Emilie A.G. Molins, Vivaswath S. Ayyar

2020Drug Metabolism and Disposition20 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryPlasma protein bindingBinding siteFree fractionDilutionSerial dilutionDrugBiophysicsBiochemistryPharmacologyBiologyThermodynamicsMedicineAlternative medicinePathologyPhysicsDrug Transport and Resistance MechanismsPharmacogenetics and Drug MetabolismPharmacological Effects and Toxicity Studies
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