Benzylaminofentanyl derivates: Discovery of bifunctional μ opioid and σ1 receptor ligands as novel analgesics with reduced adverse effects
Tao Zhuang, Jiaying Xiong, Ren Xia, Lingzhi Liang, Zhaoyang Qi, Shuang Zhang, Wei Du, Yin Chen, Xin Liu, Guisen Zhang
Topics & Concepts
ChemistryPharmacologyED50(+)-NaloxoneAntagonistAnalgesicOpioidAntagonismAgonistOpioid receptorMorphineNeuropathic painReceptorStereochemistryMedicineBiochemistryPharmacological Receptor Mechanisms and EffectsNeuropeptides and Animal PhysiologyReceptor Mechanisms and Signaling