Synthesis and antileukemic activity of an ursolic acid derivative: A potential co-drug in combination with imatinib
Elenilson Figueiredo da Silva, Artur S. de Vargas, Júlia Biz Willig, Cristiane Bernardes de Oliveira, Aline Rigon Zimmer, Diogo André Pilger, Andréia Buffon, Simone Cristina Baggio Gnoatto
Topics & Concepts
Ursolic acidMyeloid leukemiaLeukemiaPharmacologyK562 cellsBetulinic acidApoptosisChemistryImatinibCancer researchMedicineBiologyImmunologyBiochemistryGeneticsChromatographyNatural product bioactivities and synthesisRetinoids in leukemia and cellular processesToxin Mechanisms and Immunotoxins