Discovery of 3-aryl substituted benzoxaboroles as broad-spectrum inhibitors of serine- and metallo-β-lactamases
Yu‐Hang Yan, Zhaofeng Li, Xiang-Li Ning, Ji Deng, Junlin Yu, Yubin Luo, Zhenling Wang, Li Guo, Li Guo, Guo‐Bo Li, Guo‐Bo Li, You‐Cai Xiao
Topics & Concepts
ChemistryBroad spectrumSerineArylEnzymeMeropenemLactamIC50StereochemistryCarboxamideAntibioticsPharmacologyAntibiotic resistanceMicrobiologyBiochemistryIn vitroCombinatorial chemistryBiologyOrganic chemistryAlkylAntibiotic Resistance in BacteriaPneumocystis jirovecii pneumonia detection and treatmentAntimicrobial Resistance in Staphylococcus