Design, synthesis, and pharmacological evaluations of pyrrolo[1,2-a]quinoxaline-based derivatives as potent and selective sirt6 activators
Jimin Xu, Shuizhen Shi, Gang Liu, Xuping Xie, Jun Li, Andrew A. Bolinger, Haiying Chen, Wenbo Zhang, Pei‐Yong Shi, Hua Liu, Jia Zhou
Topics & Concepts
ChemistryQuinoxalineProinflammatory cytokineCytotoxicityDocking (animal)PharmacologyChemokineStereochemistryBiochemistryInflammationIn vitroImmunologyBiologyReceptorOrganic chemistryMedicineNursingSirtuins and Resveratrol in MedicinePARP inhibition in cancer therapyCalcium signaling and nucleotide metabolism