Discovery of pyrrolo[2,3-d]pyrimidine derivatives as potent Axl inhibitors: Design, synthesis and biological evaluation
Dandan Xu, Deqiao Sun, Wei Wang, Xia Peng, Zhengsheng Zhan, Yinchun Ji, Yanyan Shen, Meiyu Geng, Jing Ai, Wenhu Duan
Topics & Concepts
ChemistryPyrimidinePyrimidine analogueLead compoundPharmacologyMetastasisDrugStereochemistryCancerIn vitroBiochemistryInternal medicineBiologyMedicinePhagocytosis and Immune Regulation