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Assessment of the rat acute oral toxicity of quinoline-based pharmaceutical scaffold molecules using QSTR, q-RASTR and machine learning methods

Jianing Xu, Ting Ren, Feifan Li, Shuo Chen, Tengjiao Fan, Lijiao Zhao, Rugang Zhong, Guohui Sun, Ning Lin

2025Molecular Diversity9 citationsDOI

Topics & Concepts

QuinolineScaffoldChemistryMoleculeCombinatorial chemistryAcute toxicityToxicityStereochemistryPharmacologyOrganic chemistryComputer scienceMedicineDatabaseComputational Drug Discovery MethodsMetabolomics and Mass Spectrometry Studies