Induced expression of P-gp and BCRP transporters on brain endothelial cells using transferrin functionalized nanostructured lipid carriers: A first step of a potential strategy for the treatment of Alzheimer’s disease
Ilaria Arduino, Rosa Maria Iacobazzi, Chiara Riganti, Angela Lopedota, Maria Grazia Perrone, Antonio Lopalco, Annalisa Cutrignelli, Mariangela Cantore, Valentino Laquintana, Massimo Franco, Nicola Antonio Colabufo, Gert Luurtsema, Marialessandra Contino, Nunzio Denora
Topics & Concepts
Abcg2Blood–brain barrierTransferrin receptorTransporterTransferrinProgenitor cellEffluxStem cellPharmacologyChemistryNeural stem cellP-glycoproteinCell biologyIn vitroBiologyBiochemistryATP-binding cassette transporterMultiple drug resistanceCentral nervous systemEndocrinologyAntibioticsGeneDrug Transport and Resistance MechanismsNanoparticle-Based Drug DeliveryPharmacological Effects and Toxicity Studies