Litcius/Paper detail

Intramolecular Hydrogen Atom Transfer Hydroarylation of Alkenes toward δ-Lactams Using Cobalt-Photoredox Dual Catalysis

Yuto Yamaguchi, Yusuke Seino, Akihiko Suzuki, Yuji Kamei, Tatsuhiko Yoshino, M. Kojima, Shigeki Matsunaga

2022Organic Letters42 citationsDOIOpen Access PDF

Abstract

Intramolecular hydroarylation of alkenes through hydrogen atom transfer (HAT) represents a robust method to prepare benzo-fused heterocycles. However, the reported methods have limitations in a variety of accessible cyclic scaffolds. Here we report a dual cobalt- and photoredox-catalyzed HAT hydroarylation of alkenes that is characterized by higher efficiency in the synthesis of a δ-lactam compared to established protocols. The proposed mechanism is supported by experiments and DFT calculations.

Topics & Concepts

Intramolecular forceChemistryCobaltHydrogen atomCatalysisCombinatorial chemistryPhotochemistryStereochemistryOrganic chemistryGroup (periodic table)Catalytic C–H Functionalization MethodsRadical Photochemical ReactionsSynthesis and Catalytic Reactions