Discovery of soluble epoxide hydrolase inhibitors through DNA-encoded library technology (ELT)
Yun Ding, Svetlana Belyanskaya, Jennifer L. DeLorey, Jeffrey A. Messer, G. Joseph Franklin, Barry A. Morgan, Matthew Clark, Steven R. Skinner, Jason W. Dodson, Peng Li, Joseph P. Marino, David I. Israel
Topics & Concepts
ChemistryEpoxide hydrolase 2ChemotypeStereochemistryQuinolineEtherTriazineArylPiperidineBiochemistryEnzymeOrganic chemistryEssential oilAlkylChromatographyEicosanoids and Hypertension PharmacologyChemical Reaction MechanismsOrganic Chemistry Cycloaddition Reactions