Design, synthesis and biological evaluation of 7-((7H-pyrrolo[2,3-d]pyrimidin-4-yl)oxy)-2,3-dihydro-1H-inden-1-one derivatives as potent FAK inhibitors for the treatment of ovarian cancer
Wei Wei, Zhanzhan Feng, Zhihao Liu, Xinyue Li, Hualong He, Kai Ran, Yao Shi, Yongxia Zhu, Tinghong Ye, Chao Gao, Ningyu Wang, Luoting Yu
Topics & Concepts
ChemistryFocal adhesionIn vivoCancer researchSignal transductionIn vitroIntracellularOvarian cancerKinasePhosphorylationPharmacologyCell biologyCancerBiochemistryInternal medicineBiologyMedicineBiotechnologyCell Adhesion Molecules ResearchProtease and Inhibitor MechanismsUbiquitin and proteasome pathways