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Structural basis of SARM1 activation, substrate recognition, and inhibition by small molecules

Yun Shi, Philip S. Kerry, Jeffrey D. Nanson, Todd Bosanac, Yo Sasaki, Raul Krauss, Forhad Karim Saikot, Sarah E. Adams, Tamim Mosaiab, Veronika Masic, Xianrong Mao, Faith J. Rose, Eduardo Vasquez, Marieke Furrer, Katie Cunnea, Andrew Brearley, Weixi Gu, Zhenyao Luo, Lou Brillault, Michael J. Landsberg, Aaron DiAntonio, Boštjan Kobe, Jeffrey Milbrandt, Robert Hughes, Thomas Ve

2022Molecular Cell142 citationsDOIOpen Access PDF

Topics & Concepts

BiologySmall moleculeCell biologySubstrate specificitySubstrate (aquarium)Computational biologyBiophysicsBiochemistryEnzymeEcologyEndoplasmic Reticulum Stress and DiseaseEnzyme Structure and FunctionProtein Structure and Dynamics
Structural basis of SARM1 activation, substrate recognition, and inhibition by small molecules | Litcius