Identification of non-ATP-competitive α-carboline inhibitors of the anaplastic lymphoma kinase
Luca Mologni, Alexandre Orsato, Alfonso Zambon, Sébastien Tardy, William H. Bisson, Cédric Schneider, Monica Ceccon, Michela Viltadi, Joseph D’Attoma, Sara Pannilunghi, Vito Vece, David Gueyrard, Jerome Bertho, Léonardo Scapozza, Peter G. Goekjian, Carlo Gambacorti‐Passerini
Topics & Concepts
Anaplastic lymphoma kinaseChemistryMutantEnzymeKinaseALK inhibitorLymphomaCancer researchDrug discoveryDrugPharmacologyBiochemistryBiologyMedicineGenePleural effusionSurgeryMalignant pleural effusionImmunologyCancer therapeutics and mechanismsSynthesis and Biological EvaluationSynthesis and bioactivity of alkaloids