The Skeletal Muscle Relaxer Cyclobenzaprine Is a Potent Non-Competitive Antagonist of Histamine H1 Receptors
Kirti Singh, Ilya S. Senatorov, Ameneh Cheshmehkani, Priyanka F. Karmokar, Nader H. Moniri
Topics & Concepts
ChemistryPharmacologySkeletal muscleHistamine H1 receptorHistamineAntagonistTricyclicMuscle relaxantMuscle relaxationDiphenhydramineMuscle contractionReceptorAmitriptylineCompetitive antagonistAntagonismCurareTrachealis muscleMechanism of actionBiogenic amineAnesthesiaHistamine H2 receptorHistamine H3 receptorMast cells and histamineCoagulation, Bradykinin, Polyphosphates, and AngioedemaOlfactory and Sensory Function Studies