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Mechanistic plasticity in ApmA enables aminoglycoside promiscuity for resistance

Emily Bordeleau, P.J. Stogios, E. Evdokimova, Kalinka Koteva, Alexei Savchenko, Gerard D. Wright

2023Nature Chemical Biology10 citationsDOI

Topics & Concepts

Active siteEnzymeBiologyHistidineBiochemistryAminoglycosideChemistryGeneticsComputational biologyAntibioticsAntibiotic Resistance in BacteriaHIV/AIDS drug development and treatmentBiochemical and Molecular Research
Mechanistic plasticity in ApmA enables aminoglycoside promiscuity for resistance | Litcius