The Pharmacokinetics, Metabolism, and Clearance Mechanisms of Ritlecitinib, a Janus Kinase 3 and Tyrosine-Protein Kinase Family Inhibitor, in Humans
Jonathan Bauman, Angela C. Doran, Gabrielle M. Gualtieri, Brian Hee, Timothy J. Strelevitz, Matthew A. Cerny, Christopher Banfield, Anna Plotka, Xiaoxing Wang, Vivek S. Purohit, Martin E. Dowty
Topics & Concepts
ChemistryPharmacologyPharmacokineticsCYP2C8MetaboliteVolume of distributionTyrosine-kinase inhibitorMetabolismBioavailabilityGlutathioneCYP1A2CYP3ACytochrome P450BiochemistryCYP3A4Internal medicineEnzymeBiologyMedicineCancerColorectal Cancer Treatments and StudiesHair Growth and DisordersAutoimmune Bullous Skin Diseases