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Importance of asparagine-381 and arginine-487 for substrate recognition in CYP4Z1

Wei Du, David Machalz, Yan Qi, Erik J. Sorensen, Gerhard Wolber, Matthias Bureik

2020Biochemical Pharmacology22 citationsDOI

Topics & Concepts

AsparaginePharmacophoreSubstrate (aquarium)Binding siteEnzymeBiochemistryChemistryMutantIn silicoSubstrate specificityComputational biologyStereochemistryBiologyGeneEcologyPharmacogenetics and Drug MetabolismReceptor Mechanisms and SignalingComputational Drug Discovery Methods
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