Identification of 2-hydroxybenzoic acid derivatives as selective SIRT5 inhibitors
Yanghan Liu, Bikash Debnath, Surinder Kumar, David B. Lombard, Nouri Neamati
Topics & Concepts
ChemistrySirtuinLead compoundBiochemistryEnzymePotencyHigh-throughput screeningCarboxylic acidCombinatorial chemistryStereochemistryIn vitroNAD+ kinaseSirtuins and Resveratrol in MedicineCalcium signaling and nucleotide metabolismTea Polyphenols and Effects