Recent advances in structural types and medicinal chemistry of PARP-1 inhibitors
Ling Yu, Zhiwei Yan, Youde Wang, Miao Hao, Jingyi Zhao, Chong Pang, Shuai Li
Topics & Concepts
VeliparibOlaparibPoly ADP ribose polymerasePARP inhibitorChemistryCancer researchDNA Damage RepairBreast cancerPolymeraseSynthetic lethalityCancerDNA repairMedicineDNAInternal medicineBiochemistryPARP inhibition in cancer therapyIntegrated Circuits and Semiconductor Failure AnalysisToxin Mechanisms and Immunotoxins