15-Keto-PGE2 acts as a biased/partial agonist to terminate PGE2-evoked signaling
Suzu Endo, Akiko Suganami, Keijo Fukushima, Kanaho Senoo, Yumi Araki, John W. Regan, Masato Mashimo, Yutaka Tamura, Hiromichi Fujino
Abstract
-evoked inflammation and/or maintaining homeostasis of colorectal tissues/cells functions.
Topics & Concepts
Prostaglandin E2 receptorProstanoidReceptorAgonistAdenylyl cyclaseProstaglandinProstaglandin E2ChemistryCell biologySignal transductionEndocrinologyInternal medicineBiologyBiochemistryMedicineInflammatory mediators and NSAID effectsEstrogen and related hormone effectsEicosanoids and Hypertension Pharmacology