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Butyrolactol A enhances caspofungin efficacy via flippase inhibition in drug-resistant fungi

Xuefei Chen, H. Diessel Duan, Michael J. Hoy, Kalinka Koteva, Michaela Spitzer, Allison K. Guitor, Emily Puumala, Aline A. Fiebig, Guanggan Hu, Bonnie Yiu, Sommer Chou, Zhuyun Bian, Yeseul Choi, Amelia Bing Ya Guo, Wenliang Wang, S. Sun, Nicole Robbins, Anna Floyd Averette, Michael A. Cook, Ray Truant, Lesley T. MacNeil, Eric D. Brown, James W. Kronstad, Brian K. Coombes, Leah E. Cowen, Joseph Heitman, Huilin Li, Gerard D. Wright

2025Cell6 citationsDOIOpen Access PDF

Topics & Concepts

FlippaseEchinocandinsCaspofunginBiologyEchinocandinCryptococcus neoformansMicrobiologyBiochemistryNatural productFungal proteinPhospholipidCell biologyBiofilmAntifungalLipid IIAnidulafunginIminosugarMicrotubulePhosphatidylserineFungal growthDrug discoveryAllosteric regulationCryptococcusFungal Infections and StudiesAntifungal resistance and susceptibilityMicrobial Natural Products and Biosynthesis
Butyrolactol A enhances caspofungin efficacy via flippase inhibition in drug-resistant fungi | Litcius