Design, synthesis, biological activity evaluation and in silico studies of new nicotinohydrazide derivatives as multi-targeted inhibitors for Alzheimer's disease
Fatih Tok, Begüm Nurpelin Sağlık, Yusuf Özkay, Zafer Asım Kaplancıklı, Bedia Koçyiğit‐Kaymakçıoğlu
Topics & Concepts
ChemistrySubstituentAchéAcetylcholinesteraseIC50StereochemistryEnzymeDocking (animal)Lead compoundActive siteIn silicoCombinatorial chemistryAmyloid betaIn vitroBiochemistryPeptideGeneNursingMedicineCholinesterase and Neurodegenerative DiseasesComputational Drug Discovery MethodsAlzheimer's disease research and treatments