Discovery and development of palmatine analogues as anti-NASH agents by activating farnesoid X receptor (FXR)
Na Zhang, Tianyun Fan, Liping Zhao, Yiming Li, Yunyang Bao, Xican Ma, Yuheng Mei, Yanxiang Wang, Yonghua Liu, Hongbin Deng, Yinghong Li, Hongwei He, Danqing Song
Topics & Concepts
Farnesoid X receptorChemistryPalmatinePharmacologyIn vivoFibrosisIC50Internal medicineBiochemistryIn vitroNuclear receptorMedicineTranscription factorBiologyBiotechnologyBerberineGeneProtein Kinase Regulation and GTPase SignalingCytokine Signaling Pathways and InteractionsPI3K/AKT/mTOR signaling in cancer