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Function-oriented synthesis of Imidazo[1,2-a]pyrazine and Imidazo[1,2-b]pyridazine derivatives as potent PI3K/mTOR dual inhibitors

Chuchu Li, Yuqiao Han, Zhengyang Wang, Yanan Yu, Chen Wang, Ziwei Ren, Yanzhi Guo, Tong Zhu, XuWen Li, Suzhen Dong, Ming‐Liang Ma

2022European Journal of Medicinal Chemistry16 citationsDOIOpen Access PDF

Topics & Concepts

PI3K/AKT/mTOR pathwayChemistryIn vivoPyrazinePyridazineBioavailabilityIn vitroPharmacologyProtein kinase BSignal transductionIC50KinaseBiochemistryStereochemistryBiologyBiotechnologyPI3K/AKT/mTOR signaling in cancerQuinazolinone synthesis and applicationsCancer Mechanisms and Therapy
Function-oriented synthesis of Imidazo[1,2-a]pyrazine and Imidazo[1,2-b]pyridazine derivatives as potent PI3K/mTOR dual inhibitors | Litcius