Antitumor activity, multitarget mechanisms, and molecular docking studies of quinazoline derivatives based on a benzenesulfonamide scaffold: Cell cycle analysis
Adel S. El‐Azab, Alaa A.‐M. Abdel‐Aziz, Nawaf A. Alsaif, Hamad M. Alkahtani, Mohammed M. Alanazi, Ahmad J. Obaidullah, Razan O. Eskandrani, Amal Alharbi
Topics & Concepts
ChemistryIC50QuinazolineCytotoxicityDocking (animal)ErlotinibGefitinibTyrosine kinaseEGFR inhibitorsKinasePharmacologyBiochemistryIn vitroStereochemistryEpidermal growth factor receptorSignal transductionReceptorBiologyMedicineNursingQuinazolinone synthesis and applicationsCancer therapeutics and mechanismsHER2/EGFR in Cancer Research