Design and Synthesis of “Chloropicolinate Amides and Urea Derivatives” as Novel Inhibitors for <i>Mycobacterium tuberculosis</i>
Srihari Konduri, Dodda Bhargavi, Jyothi Prashanth, Vagolu Siva Krishna, Dharmarajan Sriram, Koya Prabhakara Rao
Abstract
for future preclinical agent drug development.
Topics & Concepts
AntimycobacterialThioureaIsoniazidChemistryMycobacterium tuberculosisMinimum inhibitory concentrationUreaDocking (animal)StereochemistryRifampicinCytotoxicityCombinatorial chemistryOrganic chemistryIn vitroTuberculosisAntimicrobialBiochemistryAntibioticsPathologyMedicineNursingSynthesis and biological activityMulticomponent Synthesis of HeterocyclesPhenothiazines and Benzothiazines Synthesis and Activities