Thiazole-based analogues as potential antibacterial agents against methicillin-resistant Staphylococcus aureus (MRSA) and their SAR elucidation
Jiaojiao Guo, Zhouling Xie, Wei Ruan, Qidong Tang, Dan Qiao, Wufu Zhu
Topics & Concepts
ThiazoleStaphylococcus aureusPharmacophoreAntibioticsAntibacterial activityChemistryDrugAntibiotic resistanceDrug resistanceAntibacterial agentPharmacologyMicrobiologyCombinatorial chemistryBacteriaMedicineBiologyStereochemistryBiochemistryGeneticsSynthesis and biological activityClick Chemistry and ApplicationsQuinazolinone synthesis and applications