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PI3Kδ and mTOR dual inhibitors: Design, synthesis and anticancer evaluation of 3-substituted aminomethylquinoline analogues

Digambar Yevale, Nishith Teraiya, Twinkle Lalwani, Mayur Dalasaniya, Khushal M. Kapadiya, Rakesh Kumar Ameta, Chetan B. Sangani, Yongtao Duan

2024Bioorganic Chemistry22 citationsDOI

Topics & Concepts

PI3K/AKT/mTOR pathwayChemistryApoptosisIC50AnnexinPharmacologyBiochemistryIn vitroBiologyPI3K/AKT/mTOR signaling in cancerChronic Lymphocytic Leukemia ResearchCytokine Signaling Pathways and Interactions
PI3Kδ and mTOR dual inhibitors: Design, synthesis and anticancer evaluation of 3-substituted aminomethylquinoline analogues | Litcius