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State-Dependent Inhibition of Nav1.8 Sodium Channels by VX-150 and VX-548

Patric Vaelli, Akie Fujita, Sooyeon Jo, Han-Xiong Bear Zhang, Tomás Osorno, Xiao Ma, Bruce P. Bean

2024Molecular Pharmacology48 citationsDOIOpen Access PDF

Topics & Concepts

ChemistryIon channel regulation and functionNicotinic Acetylcholine Receptors StudyNeuroscience and Neuropharmacology Research