Structural basis of GPBAR activation and bile acid recognition
Fan Yang, Chunyou Mao, Lulu Guo, Jing‐Yu Lin, Qianqian Ming, Peng Xiao, Xiang Wu, Qingya Shen, Shimeng Guo, Dandan Shen, Ruirui Lu, Linqi Zhang, Shen-Ming Huang, Yuqi Ping, Chenlu Zhang, Cheng Ma, Kai Zhang, Xiaoying Liang, Yuemao Shen, Fajun Nan, Fan Yi, Vincent C. Luca, Jiuyao Zhou, Changtao Jiang, Jin‐Peng Sun, Xin Xie, Xiao Yu, Yan Zhang
Topics & Concepts
Allosteric regulationCholic acidBile acidG protein-coupled bile acid receptorBiochemistryBinding siteLigand (biochemistry)ChemistryMolecular recognitionProtein structureReceptorBiophysicsStereochemistryBiologyMoleculeOrganic chemistryDrug Transport and Resistance MechanismsReceptor Mechanisms and SignalingLipid Membrane Structure and Behavior