Synthesis and biological evaluation of novel pyrrolo[2,3-b]pyridine derivatives as potent GSK-3β inhibitors for treating Alzheimer's disease
Qingqing Xun, Jing Zhang, Yan-Peng Li, Ying Li, Yuying Ma, Zhaobin Chen, Le-Ping Ding, Xiao-Long Shi
Topics & Concepts
ChemistryPyridineChemical synthesisStereochemistryBiological activityCombinatorial chemistryBiochemistryIn vitroMedicinal chemistryCholinesterase and Neurodegenerative DiseasesNuclear Receptors and SignalingPhosphodiesterase function and regulation