Synthesis, and biological evaluation of 3,6-diaryl-[1,2,4]triazolo[4,3-a]pyridine analogues as new potent tubulin polymerization inhibitors
Fang Yang, Xie‐Er Jian, Peng-Cheng Diao, Xian‐Sen Huo, Wen‐Wei You, Pei‐Liang Zhao
Topics & Concepts
ChemistryTubulinStereochemistryHeLaIC50MicrotubulePolymerizationPyridineMicrotubule polymerizationCell cycleBiochemistryIn vitroApoptosisOrganic chemistryBiologyPolymerCell biologySynthesis and biological activityClick Chemistry and ApplicationsSynthesis and Biological Evaluation