Synthesis and in vitro antitrypanosomal evaluation of novel 6-heteroarylidene-substituted quinolone derivatives
Klaudia T. Angula, Lesetja J. Legoabe, Tarryn Swart, Heinrich C. Hoppe, Richard M. Beteck
Topics & Concepts
QuinoloneChemistryAfrican trypanosomiasisTrypanosoma bruceiIC50PharmacologyIn vitroIn vivoTrypanocidal agentMoietyTrypanosomiasisCombinatorial chemistryStereochemistryBiochemistryBiologyAntibioticsVirologyBiotechnologyGeneTrypanosoma species research and implicationsResearch on Leishmaniasis StudiesSynthesis and Biological Evaluation