An optimized BRD4 inhibitor effectively eliminates NF-κB-driven triple-negative breast cancer cells
Guan‐Jun Yang, Yingqi Song, Wanhe Wang, Quan‐Bin Han, Dik‐Lung Ma, Chung‐Hang Leung
Topics & Concepts
BromodomainTriple-negative breast cancerAcetylationBRD4ChemistryCancer researchNF-κBCancerBreast cancerBiochemistryBiologySignal transductionGeneticsGeneProtein Degradation and InhibitorsMultiple Myeloma Research and TreatmentsUbiquitin and proteasome pathways