Novel 6,7,8-trihydrobenzo[6',7']cyclohepta[2',1'-e]pyrazolo[2,3-a]pyrimidine derivatives as Topo IIα inhibitors with potential cytotoxic activity
Thoraya A. Farghaly, Hanan Gaber Abdulwahab, Hanadi Y. Medrasi, Mariam A. Al‐Sheikh, Dina F. Katowah, Amani M.R. Alsaedi
Topics & Concepts
ChemistryStereochemistryPyrimidineIC50DoxorubicinDocking (animal)TopoisomeraseIn vitroCytotoxicityBiochemistryChemotherapyNursingMedicineSurgeryCancer therapeutics and mechanismsSynthesis and bioactivity of alkaloidsBioactive Compounds and Antitumor Agents