Flavones reversibly inhibit Leishmania donovani tyrosine aminotransferase by binding to the catalytic pocket: An integrated in silico-in vitro approach
Santanu Sasidharan, Prakash Saudagar
Topics & Concepts
In silicoChemistryLeishmania donovaniIn vitroLeishmaniaActive sitePharmacophoreDrugElectrophileStereochemistryLipophilicityCombinatorial chemistryReactivity (psychology)Tyrosine aminotransferaseBiochemistryCatalysisEnzymeVisceral leishmaniasisLeishmaniasisPharmacologyBiologyMedicineWorld Wide WebGenePathologyParasite hostingAlternative medicineEnzyme inducerComputer scienceImmunologyResearch on Leishmaniasis StudiesTrypanosoma species research and implicationsSynthesis and biological activity