Discovery of quinazolin-4(3H)-one derivatives as novel AChE inhibitors with anti-inflammatory activities
Ling Lv, Mireguli Maimaitiming, Yan Huang, Jichen Yang, Shuxia Chen, Yanfeng Sun, Xuetao Zhang, Xin Li, Changhu Xue, Pingyuan Wang, Chang‐Yun Wang, Zhiqing Liu
Topics & Concepts
ChemistryAcetylcholinesteraseButyrylcholinesteraseAchéCholinesteraseIC50PharmacologyNeuroinflammationProinflammatory cytokineDocking (animal)Inhibitory postsynaptic potentialEnzymeStereochemistryBiochemistryIn vitroInflammationInternal medicineMedicineNursingCholinesterase and Neurodegenerative DiseasesPhenothiazines and Benzothiazines Synthesis and ActivitiesComputational Drug Discovery Methods