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Discovery of anti-neuroinflammatory agents from 1,4,5,6-tetrahydrobenzo[2,3]oxepino[4,5-d]pyrimidin-2-amine derivatives by regulating microglia polarization

Yang Yang, Zhongfei Gao, Gui‐Ge Hou, Qingguo Meng, Yun Hou

2023European Journal of Medicinal Chemistry13 citationsDOI

Topics & Concepts

MicrogliaNeuroinflammationChemistryPharmacologyLipopolysaccharideTumor necrosis factor alphaCell biologyInflammationImmunologyMedicineBiologyNeuroinflammation and Neurodegeneration MechanismsTryptophan and brain disordersImmune cells in cancer
Discovery of anti-neuroinflammatory agents from 1,4,5,6-tetrahydrobenzo[2,3]oxepino[4,5-d]pyrimidin-2-amine derivatives by regulating microglia polarization | Litcius