Isatin-Schiff's base and chalcone hybrids as chemically apoptotic inducers and EGFR inhibitors; design, synthesis, anti-proliferative activities and in silico evaluation
Eman A. Fayed, Rogy R. Ezz Eldin, Ahmed B. M. Mehany, Ashraf H. Bayoumi, Yousry A. Ammar
Topics & Concepts
IsatinChemistryChalconeIC50ApoptosisCell cultureLapatinibPharmacologyIn silicoErlotinibCytotoxicityStereochemistryBiochemistryIn vitroCancerEpidermal growth factor receptorReceptorOrganic chemistryGeneticsTrastuzumabBiologyInternal medicineBreast cancerGeneMedicineSynthesis and biological activitySynthesis and Characterization of Heterocyclic CompoundsQuinazolinone synthesis and applications