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A new class of cytotoxic agents targets tubulin and disrupts microtubule dynamics

Ayad A. Al-Hamashi, Radhika Koranne, Samkeliso Dlamini, Abdulateef Alqahtani, Endri Karaj, Maisha S. Rashid, Joseph R. Knoff, Matthew Dunworth, Mary Kay H. Pflum, Robert A. Casero, L. Perera, William R. Taylor, L. M. Viranga Tillekeratne

2021Bioorganic Chemistry19 citationsDOIOpen Access PDF

Topics & Concepts

TubulinChemistryMitosisMicrotubule polymerizationMicrotubuleMechanism of actionDocking (animal)BiochemistryCytotoxicityCancer cellNocodazoleChalconeCell biologyIn vitroStereochemistryCellBiologyCytoskeletonCancerNursingGeneticsMedicineHistone Deacetylase Inhibitors ResearchProtein Degradation and InhibitorsCancer Mechanisms and Therapy
A new class of cytotoxic agents targets tubulin and disrupts microtubule dynamics | Litcius