Discovery and computational studies of 2-phenyl-benzoxazole acetamide derivatives as promising P2Y14R antagonists with anti-gout potential
Mengze Zhou, Weiwei Wang, Zhongkui Wang, Yilin Wang, Yifan Zhu, Zhiqian Lin, Sheng Tian, Yuan Huang, Qinghua Hu, Huanqiu Li
Topics & Concepts
BenzoxazoleChemistryAcetamideIn vivoPharmacologyGoutAntagonistLead compoundIC50Virtual screeningArthritisDocking (animal)Ex vivoReceptorStereochemistryIn vitroBiochemistryDrug discoveryMedicineInternal medicineBiotechnologyBiologyOrganic chemistryNursingAdenosine and Purinergic SignalingUrticaria and Related ConditionsNeuropeptides and Animal Physiology