Litcius/Paper detail

Antibiotic Conjugates with an Artificial MECAM-Based Siderophore Are Potent Agents against Gram-Positive and Gram-Negative Bacterial Pathogens

Lukas Pinkert, Yi-Hui Lai, Carsten Peukert, Sven‐Kevin Hotop, Bianka Karge, Lara Marie Schulze, Jörg Grunenberg, Mark Brönstrup

2021Journal of Medicinal Chemistry52 citationsDOIOpen Access PDF

Abstract

was mediated by a mutation in the gene encoding ExbB, which is involved in siderophore transport.

Topics & Concepts

SiderophoreEscherichia coliChemistryMicrobiologyIn silicoDaptomycinBacteriaAntibioticsGram-negative bacteriaBacterial outer membraneAntimicrobialLinkerMutantAntibiotic resistanceConjugateGram-positive bacteriaBiochemistryBiologyGeneStaphylococcus aureusOperating systemMathematicsComputer scienceMathematical analysisGeneticsVancomycinAntibiotic Resistance in BacteriaBacterial Genetics and BiotechnologyCancer therapeutics and mechanisms