Litcius/Paper detail

Targeting protein conformations with small molecules to control protein complexes

Emmanouil Zacharioudakis, Evripidis Gavathiotis

2022Trends in Biochemical Sciences19 citationsDOIOpen Access PDF

Topics & Concepts

Small moleculeDrug discoveryRational designProtein functionChemistryFunction (biology)Protein–protein interactionComputational biologyProtein structureBiophysicsBiochemistryCell biologyBiologyGeneGeneticsUbiquitin and proteasome pathways14-3-3 protein interactionsRNA and protein synthesis mechanisms