Structural optimization towards promising β-methyl-4-acrylamido quinoline derivatives as PI3K/mTOR dual inhibitors for anti-cancer therapy: The in vitro and in vivo biological evaluation
Ruoyu He, Bingyong Xu, Ping Li, Xiaoqing Lv
Topics & Concepts
PI3K/AKT/mTOR pathwayChemistryIn vivoCmaxPharmacologyKinaseIn vitroBiochemistrySignal transductionBioavailabilityMedicineBiologyBiotechnologyPI3K/AKT/mTOR signaling in cancerTuberous Sclerosis Complex ResearchChronic Myeloid Leukemia Treatments